Browsing Universitätsbibliographie by Author "Koch, Pierre"

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2-Alkylsulfanyl-4(5)-aryl-5(4)-heteroarylimidazoles: An Overview on Synthetic Strategies and Biological Activity

Koch, Pierre; Ansideri, Francesco (2017)
A Diverse and Versatile Regiospecific Synthesis of Tetrasubstituted Alkylsulfanylimidazoles as p38 Mitogen-Activated Protein Kinase Inhibitors

Ansideri, Francesco; Andreev, Stanislav; Kuhn, Annette; Albrecht, Wolfgang; Laufer, Stefan A.; Koch, Pierre (2018)
A novel LysR-type regulator negatively affects biosynthesis of the immunosuppressant brasilicardin

Wolanski, Marcin; Krawiec, Michal; Schwarz, Paul N.; Stegmann, Evi; Wohlleben, Wolfgang; Buchmann, Anina; Gross, Harald; Eitel, Michael; Koch, Pierre; Botas, Alma; Mendez, Carmen; Elena Nunez, Luz; Moris, Francisco; Cortes, Jesus; Zakrzewska-Czerwinska, Jolanta (2021)
Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3 beta Inhibitors

Andreev, Stanislav; Pantsar, Tatu; Tesch, Roberta; Kahlke, Niclas; El-Gokha, Ahmed; Ansideri, Francesco; Graetz, Lukas; Romasco, Jenny; Sita, Giulia; Geibel, Christian; Laemmerhofer, Michael; Tarozzi, Andrea; Knapp, Stefan; Laufer, Stefan A.; Koch, Pierre (2022)
An optimized and versatile synthesis to pyridinylimidazole-type p38 alpha mitogen activated protein kinase inhibitors

El-Gokha, Ahmed; Laufer, Stefan A.; Koch, Pierre (2015)
c-Jun N-terminal kinase inhibitors: a patent review (2010-2014)

Gehringer, Matthias; Muth, Felix; Koch, Pierre; Laufer, Stefan A. (2015)
Design and Synthesis of Highly Selective Brain Penetrant p38 alpha Mitogen-Activated Protein Kinase Inhibitors

Tormaehlen, Niklas M.; Martorelli, Mariella; Kuhn, Annette; Maier, Florian; Guezguez, Jamil; Burnet, Michael; Albrecht, Wolfgang; Laufer, Stefan A.; Koch, Pierre (2022)
Design, Synthesis and Biological Evaluation of 7-Chloro-9H-pyrimido[4,5-b]indole-based Glycogen Synthase Kinase-3 beta Inhibitors

Andreev, Stanislav; Pantsar, Tatu; Ansideri, Francesco; Kudolo, Mark; Forster, Michael; Schollmeyer, Dieter; Laufer, Stefan A.; Koch, Pierre (2019)
Discovery and Evaluation of Enantiopure 9H-pyrimido[4,5-b]indoles as Nanomolar GSK-3 beta Inhibitors with Improved Metabolic Stability

Andreev, Stanislav; Pantsar, Tatu; El-Gokha, Ahmed; Ansideri, Francesco; Kudolo, Mark; Anton, Debora Bublitz; Sita, Giulia; Romasco, Jenny; Geibel, Christian; Laemmerhofer, Michael; Goettert, Marcia Ines; Tarozzi, Andrea; Laufer, Stefan A.; Koch, Pierre (2020)
Evaluation of Novel Substituted Furopyridines as Inhibitors of Protein Kinases Related to Tau Pathology in Alzheimer's Disease

Schade, N.; Koch, P.; Ansideri, F.; Krystof, V.; Holzer, M.; Hilgeroth, A. (2021)
Fluorescence polarization-based assays for detecting compounds binding to inactive c-Jun N-terminal kinase 3 and p38 alpha mitogen-activated protein kinase

Ansideri, Francesco; Lange, Andreas; El-Gokha, Ahmed; Boeckler, Frank M.; Koch, Pierre (2016)
Fluorescence polarization-based competition binding assay for c-Jun N-terminal kinases 1 and 2

Ansideri, Francesco; Dammann, Marcel; Boeckler, Frank M.; Koch, Pierre (2017)
From 2-Alkylsulfanylimidazoles to 2-Alkylimidazoles: An Approach towards Metabolically More Stable p38 alpha MAP Kinase Inhibitors

Heider, Fabian; Haun, Urs; Doering, Eva; Kudolo, Mark; Sessler, Catharina; Albrecht, Wolfgang; Laufer, Stefan; Koch, Pierre (2017)
Genetic Engineering in Combination with Semi-Synthesis Leads to a New Route for Gram-Scale Production of the Immunosuppressive Natural Product Brasilicardin A

Botas, Alma; Eitel, Michael; Schwarz, Paul N.; Buchmann, Anina; Costales, Paula; Nunez, Luz Elena; Cortes, Jesus; Moris, Francisco; Krawiec, Michal; Wolanski, Marcin; Gust, Bertolt; Rodriguez, Mirna; Fischer, Wolf-Nicolas; Jandeleit, Bernd; Zakrzewska-Czerwinska, Jolanta; Wohlleben, Wolfgang; Stegmann, Evi; Koch, Pierre; Mendez, Carmen; Gross, Harald (2021)
Halogen-enriched fragment libraries as chemical probes for harnessing halogen bonding in fragment-based lead discovery

Zimmermann, Markus O.; Lange, Andreas; Wilcken, Rainer; Cieslik, Markus B.; Exner, Thomas E.; Joerger, Andreas C.; Koch, Pierre; Boeckler, Frank M. (2014)
Inhibitors of c-Jun N-Terminal Kinases: An Update

Koch, Pierre; Gehringer, Matthias; Laufer, Stefan A. (2015)
Probing Substituents in the 1-and 3-Position : Tetrahydropyrazino-Annelated Water-Soluble Xanthine Derivatives as Multi-Target Drugs With Potent Adenosine Receptor Antagonistic Activity

Koch, Pierre; Brunschweiger, Andreas; Namasivayam, Vigneshwaran; Ullrich, Stefan; Maruca, Annalisa; Lazzaretto, Beatrice; Kueppers, Petra; Hinz, Sonja; Hockemeyer, Joerg; Wiese, Michael; Heer, Jag; Alcaro, Stefano; Kiec-Kononowicz, Katarzyna; Mueler, Christa E. (2018)
Pyridinylimidazoles as dual glycogen synthase kinase 3 beta/p38 alpha mitogen-activated protein kinase inhibitors

Heider, Fabian; Ansideri, Francesco; Tesch, Roberta; Pantsar, Tatu; Haun, Urs; Doering, Eva; Kudolo, Mark; Poso, Antti; Albrecht, Wolfgang; Laufer, Stefan A.; Koch, Pierre (2019)
Pyridinylimidazoles as GSK3 beta Inhibitors: The Impact of Tautomerism on Compound Activity via Water Networks

Heider, Fabian; Pantsar, Tatu; Kudolo, Mark; Ansideri, Francesco; De Simone, Angela; Pruccoli, Letizia; Schneider, Taiane; Goettert, Marcia Ines; Tarozzi, Andrea; Andrisano, Vincenza; Laufer, Stefan A.; Koch, Pierre (2019)
Selective mono-de-O-acetylation of the per-O-acetylated brasilicardin carbohydrate side chain

Eitel, Michael; Zinad, Dhafer S.; Schollmeyer, Dieter; Gross, Harald; Koch, Pierre (2021)

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